Setiptiline maleate is a tetracyclic antidepressant (TeCA) that functions as a noradrenergic and specific serotonergic antidepressant (NaSSA). It acts as a norepinephrine reuptake inhibitor and an α2-adrenergic receptor antagonist, as well as a serotonin receptor antagonist, likely affecting the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes. It also functions as an H1 receptor inverse agonist/antihistamine, making it suitable for research applications.
- High purity (99.94%) for reliable research
- Well-characterized pharmacological actions
- Inhibits norepinephrine reuptake
- Antagonizes α2-adrenergic receptors
- Antagonizes serotonin receptors (5-HT2A, 5-HT2C, and/or 5-HT3)
- Acts as an H1 receptor inverse agonist/antihistamine
- Detailed solubility information and protocols for in vitro and in vivo studies